| Product Number : |
CL2754 |
| Product Name : |
BIX-01294 |
| CAS No. : |
935693-62-2 |
| Synonyms : |
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| Chemical Name : |
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| Molecular Formula : |
C28H38N6O2 |
| Molecular Weight : |
490.64 |
| Molecular Structure : |
 |
| Appearance : |
White to off-white powder |
| Specification : |
98+% |
| Application : |
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| Registration : |
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| Storage Condition : |
BIX-01294 is a reversible and highly selective G9a and GLP Histone Methyltransferase inhibitor, with IC50s of of 1.7 μM and 0.9 μM, respectively. BIX-01294 inhibits G9a/GLP by competing for binding with the amino acids N-terminal of the substrate lysine residue. BIX-01294, a (1H-1,4-diazepin-1-yl)-quinazolin-4-yl amine derivative, induces necroptosis and autophagy. BIX-01294 has antitumor activity in recurrent tumor cells
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->>Products covered by valid patents are not offered or supplied for commercial use.
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->>Any patent infringement and resulting liability is solely at buyer's risk.
->>Our products are only raw materials for drugs or industry, can't be used for human or animals directly.
